01423nam a22001457a 4500008004100000020001800041050001400059100001800073245017700091250001200268260004500280300003400325500002000359505089800379151029b xxu||||| |||| 00| 0 eng d a9788122430868 aRS403.K37 aKar, Ashutosh aMedicinal chemistry: introduction - classification - synthesis - explanation - mechanism of action - structure activity relationships (SARs) - usages - doses.cAshutosh Kar a5th ed. aNew Delhi:bNew Age Techno Press,c2010. axxvi, 1013p.:bills.;c25 cm. aIncludes index. aContent: Drug design - A rational approach -- Physical-chemical factors and biological activities -- Molecular modelling and design -- General anaesthetics -- Local anaesthetics -- Sedatives and hypnotics -- Anticonvulsants -- Muscle relaxants -- Central nervous system stimulants -- Antipyretic analgesics -- Narcotic analgesics (opiate analgesics) -- Cardiovascular drugs -- Autonomic drugs -- Diuretics -- Antihistamincs -- Non-steroidal anti-inflammatory drugs (NSAIDs) -- Antiparkinsonism agents -- Expectorants and antitussives -- Sulphonamides -- Antimalarials -- Anthelmintics -- Insulin and oral hypoglycemic agents -- Steroids -- Adrenocortal steroids -- Antibiotics -- Antimycobacterial drugs -- Antineoplastic agents -- Antipsychotics (tranquilizers) -- Antiviral drugs -- Newer drugs for newer diseases -- Pro-drug approach in drug design -- Drug discovery via enzyme inhibition.